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204
"Further insights of selenium-containing analogues of WC-9 against Trypanosoma cruzi" (2019) Chao, M.N.;Lorenzo-Ocampo, M.V.;Szajnman, S.H. (...)Rodriguez, J.B. Bioorganic and Medicinal Chemistry. 27(7):1350-1361
"Synthesis and biological evaluation of new quinoline derivatives as antileishmanial and antitrypanosomal agents" (2019) Chanquia, S.N.;Larregui, F.;Puente, V. (...)García Liñares, G. Bioorganic Chemistry. 83:526-534
"Synthesis, molecular docking and biological evaluation of novel phthaloyl derivatives of 3-amino-3-aryl propionic acids as inhibitors of Trypanosoma cruzi trans-sialidase" (2018) Kashif, M.;Chacón-Vargas, K.F.;López-Cedillo, J.C. (...)Rivera, G. European Journal of Medicinal Chemistry. 156:252-268
"Lipophilic Decyl Chain-Pterin Conjugates with Sensitizer Properties" (2018) Vignoni, M.;Walalawela, N.;Bonesi, S.M. (...)Thomas, A.H. Molecular Pharmaceutics. 15(3):798-807
"Synthesis and activity evaluation of a series of cholanamides as modulators of the liver X receptors" (2018) Martínez, M.D.;Ghini, A.A.;Dansey, M.V. (...)Burton, G. Bioorganic and Medicinal Chemistry. 26(5):1092-1101
"Chemoenzymatic synthesis of new derivatives of glycyrrhetinic acid with antiviral activity. Molecular docking study" (2018) Zígolo, M.A.;Salinas, M.;Alché, L. (...)Liñares, G.G. Bioorganic Chemistry. 78:210-219
"Oxidation at C-16 enhances butyrylcholinesterase inhibition in lupane triterpenoids" (2018) Castro, M.J.; Richmond, V.; Faraoni, M.B.; Murray, A.P. Bioorganic Chemistry. 79:301-309
"Dimerization, redox properties and antioxidant activity of two manganese(III) complexes of difluoro- and dichloro-substituted Schiff-base ligands" (2017) Palopoli, C.;Gómez, G.;Foi, A. (...)Signorella, S. Journal of Inorganic Biochemistry. 167:49-59
"Synthesis of new C-25 and C-26 steroidal acids as potential ligands of the nuclear receptors DAF-12, LXR and GR" (2017) Dansey, M.V.; del Fueyo, M.C.; Veleiro, A.S.; Di Chenna, P.H. Steroids. 121:40-46
"Synthesis and cytotoxicity evaluation of A-ring derivatives of cycloartanone" (2017) Zambrano, E.E.;Casas, A.G.;Di Venosa, G.M. (...)Palermo, J.A. Phytochemistry Letters. 21:200-205
"Synthesis and in vitro antiproliferative activities of (5-aryl-1,2,4-oxadiazole-3-yl) methyl D-ribofuranosides" (2017) Avanzo, R.E.; Padrón, J.M.; D'Accorso, N.B.; Fascio, M.L. Bioorganic and Medicinal Chemistry Letters. 27(16):3674-3677
"Selenium-containing analogues of WC-9 are extremely potent inhibitors of Trypanosoma cruzi proliferation" (2017) Chao, M.N.;Storey, M.;Li, C. (...)Rodriguez, J.B. Bioorganic and Medicinal Chemistry. 25(24):6435-6449
"Synthesis and antifungal activity of bile acid-derived oxazoles" (2016) Fernández, L.R.;Svetaz, L.;Butassi, E. (...)Sánchez, M. Steroids. 108:68-76
"Synthetic stigmastanes with dual antiherpetic and immunomodulating activities inhibit ERK and Akt signaling pathways without binding to glucocorticoid receptors" (2016) Michelini, F.M.;Bueno, C.A.;Molinari, A.M. (...)Ramírez, J.A. Biochimica et Biophysica Acta - General Subjects. 1860(1):129-139
"Anti-hemagglutinin antibody derived lead peptides for inhibitors of influenza virus binding" (2016) Memczak, H.;Lauster, D.;Kar, P. (...)Stöcklein, W.F.M. PLoS ONE. 11(7)
"Synthetic pregnenolone derivatives as antiviral agents against acyclovir-resistant isolates of Herpes Simplex Virus Type 1" (2015) Dávola, M.E.;Mazaira, G.I.;Galigniana, M.D. (...)Barquero, A.A. Antiviral Research. 122:55-63
"Imidazothiazole and related heterocyclic systems. Synthesis, chemical and biological properties" (2015) Fascio, M.L.; Errea, M.I.; D'Accorso, N.B. European Journal of Medicinal Chemistry. 90:666-683
"Lipase-catalyzed preparation of mono- and diesters of ferulic acid" (2015) Sandoval, G.;Quintana, P.G.;Baldessari, A. (...)Plou, F.J. Biocatalysis and Biotransformation. 33(2):89-97
"Aryloxyethyl thiocyanates are potent growth inhibitors of Trypanosoma cruzi and Toxoplasma gondii" (2015) Chao, M.N.;Matiuzzi, C.E.;Storey, M. (...)Rodriguez, J.B. ChemMedChem. 10(6):1094-1108
"Structure-activity relationship of hybrids of Cinchona alkaloids and bile acids with in vitro antiplasmodial and antitrypanosomal activities" (2015) Leverrier, A.;Bero, J.;Cabrera, J. (...)Palermo, J.A. European Journal of Medicinal Chemistry. 100(1):10-17
"Synthesis and biological evaluation of salpichrolide analogs as antiestrogenic agents" (2014) Sonego, J.M.;Rivero, E.M.;Gargiulo, L. (...)Burton, G. European Journal of Medicinal Chemistry. 82:233-241
"Enhancing antibacterial activity against Escherichia coli K-12 of peptide Ib-AMP4 with synthetic analogues" (2014) Flórez-Castillo, J.M.; Perullini, M.; Jobbágy, M.; De Jesús Cano Calle, H. International Journal of Peptide Research and Therapeutics. 20(3):365-369
"QSAR on antiproliferative naphthoquinones based on a conformation- independent approach" (2014) Duchowicz, P.R.;Bennardi, D.O.;Bacelo, D.E. (...)Misico, R.I. European Journal of Medicinal Chemistry. 77:176-184
"Synthesis and cholinesterase inhibition of cativic acid derivatives" (2014) Alza, N.P.;Richmond, V.;Baier, C.J. (...)Murray, A.P. Bioorganic and Medicinal Chemistry. 22(15):3838-3849
"New insights into molecular recognition of 1,1-bisphosphonic acids by farnesyl diphosphate synthase" (2014) Ferrer-Casal, M.;Li, C.;Galizzi, M. (...)Rodriguez, J.B. Bioorganic and Medicinal Chemistry. 22(1):398-405
"Synthesis and cytotoxic evaluation of four new 6E-hydroximinosteroids" (2014) Richmond, V.;Careaga, V.P.;Sacca, P. (...)Maier, M.S. Steroids. 84:7-10
"Differential effect of heterocyclic d-ribofuranoside derivatives on human prostate cancer cell viability and cell cycle progression" (2014) Gueron, G.;Avanzo, R.E.;Schuster, F. (...)D'Accorso, N.B. Biomedicine and Pharmacotherapy. 68(7):847-854
"Multicomponent synthesis of 4,4-dimethyl sterol analogues and their effect on eukaryotic cells" (2014) Alonso, F.;Cirigliano, A.M.;Dávola, M.E. (...)Ramírez, J.A. Steroids. 84:1-6
"Preparation, anticholinesterase activity and molecular docking of new lupane derivatives" (2014) Castro, M.J.;Richmond, V.;Romero, C. (...)Murray, A.P. Bioorganic and Medicinal Chemistry. 22(13):3341-3350
"Acridones as antiviral agents: Synthesis, chemical and biological properties" (2013) Sepúlveda, C.S.;Fascio, M.L.;García, C.C. (...)Damonte, E.B. Current Medicinal Chemistry. 20(19):2402-2414
"Synthesis and biological evaluation of novel substituted pyrrolo[1,2-a] quinoxaline derivatives as inhibitors of the human protein kinase CK2" (2013) Guillon, J.;Le Borgne, M.;Rimbault, C. (...)Jose, J. European Journal of Medicinal Chemistry. 65:205-222
"Design, synthesis and biological evaluation of sulfur-containing 1,1-bisphosphonic acids as antiparasitic agents" (2013) Recher, M.;Barboza, A.P.;Li, Z.-H. (...)Rodriguez, J.B. European Journal of Medicinal Chemistry. 60:431-440
"Synthesis of the (1→6)-linked thiodisaccharide of galactofuranose: Inhibitory activity against a β-galactofuranosidase" (2013) Repetto, E.; Marino, C.; Varela, O. Bioorganic and Medicinal Chemistry. 21(11):3327-3333
"Preparation and antitrypanosomal activity of secochiliolide acid derivatives" (2013) Siless, G.E.;Lozano, E.;Sánchez, M. (...)Palermo, J.A. Bioorganic and Medicinal Chemistry Letters. 23(17):4964-4967
"27-Nor-Δ4-dafachronic acid is a synthetic ligand of Caenorhabditis elegans DAF-12 receptor" (2013) Samaja, G.A.;Castro, O.;Alvarez, L.D. (...)Burton, G. Bioorganic and Medicinal Chemistry Letters. 23(10):2893-2896
"Synthesis of 6-azaprogesterone and 19-hydroxy-6-azasteroids" (2013) Martínez, M.D.;Edelsztein, V.C.;Durán, F.J. (...)Burton, G. Steroids. 78(1):34-37
"Synthesis and antifungal activity of C-21 steroids with an aromatic D ring" (2013) Sonego, J.M.;Cirigliano, A.M.;Cabrera, G.M. (...)Veleiro, A.S. Steroids. 78(7):644-650
"Antiparasitic hybrids of Cinchona alkaloids and bile acids" (2013) Leverrier, A.;Bero, J.;Frédérich, M. (...)Palermo, J. European Journal of Medicinal Chemistry. 66:355-363
"Antiparasitic hybrids of Cinchona alkaloids and bile acids" (2013) Leverrier, A.;Bero, J.;Frédérich, M. (...)Palermo, J. European Journal of Medicinal Chemistry. 66:355-363
"Chemical constituents and biological activity of euglena gracilis extracts" (2013) Tolivia, A.; Conforti, V.; Córdoba, O.; Flores, L. Journal of Pharmacy Research. 7(3):209-214
"Design, synthesis and biological evaluation of WC-9 analogs as antiparasitic agents" (2013) Elicio, P.D.;Chao, M.N.;Galizzi, M. (...)Rodriguez, J.B. European Journal of Medicinal Chemistry. 69:480-489
"β-Lapachone analogs with enhanced antiproliferative activity" (2012) Ríos-Luci, C.;Bonifazi, E.L.;León, L.G. (...)Padrón, J.M. European Journal of Medicinal Chemistry. 53:264-274
"Chemoenzymatic synthesis and biological evaluation of 2- and 3-hydroxypyridine derivatives against Leishmania mexicana" (2012) García Liñares, G.; Parraud, G.; Labriola, C.; Baldessari, A. Bioorganic and Medicinal Chemistry. 20(15):4614-4624
"Sterol analogues with diamide side chains interfere with the intracellular localization of viral glycoproteins" (2012) Dávola, M.E.;Alonso, F.;Cabrera, G.M. (...)Barquero, A.A. Biochemical and Biophysical Research Communications. 427(1):107-112
"Multicomponent synthesis of acylated short peptoids with antifungal activity against plant pathogens" (2012) Galetti, M.D.; Cirigliano, A.M.; Cabrera, G.M.; Ramírez, J.A. Molecular Diversity. 16(1):113-119
"1,2,4-Triazole d-ribose derivatives: Design, synthesis and antitumoral evaluation" (2012) Avanzo, R.E.;Anesini, C.;Fascio, M.L. (...)D'Accorso, N.B. European Journal of Medicinal Chemistry. 47(1):104-110
"Synthesis and cytotoxic activity evaluation of dihydrocucurbitacin B and cucurbitacin B derivatives" (2012) Lang, K.L.;Silva, I.T.;Zimmermann, L.A. (...)Durán, F.J. Bioorganic and Medicinal Chemistry. 20(9):3016-3030
"Synthesis and acetylcholinesterase inhibitory activity of 2β,3α-disulfoxy-5α-cholestan-6-one" (2011) Richmond, V.; Santos, G.A.G.; Murray, A.P.; Maier, M.S. Steroids. 76(10-11):1160-1165
"Synthesis of multivalent glycoclusters from 1-thio-β-D-galactose and their inhibitory activity against the β-galactosidase from E. coli" (2011) Cagnoni, A.J.;Varela, O.;Gouin, S.G. (...)Uhrig, M.L. Journal of Organic Chemistry. 76(9):3064-3077
"Imidazo[2,1-b]thiazole carbohydrate derivatives: Synthesis and antiviral activity against Junin virus, agent of Argentine hemorrhagic fever" (2011) Barradas, J.S.;Errea, M.I.;D'Accorso, N.B. (...)Damonte, E.B. European Journal of Medicinal Chemistry. 46(1):259-264
"Synthesis and biological evaluation of N-thia-carba-thymidine as an antiherpetic agent" (2010) Elhalem, E.; Pujol, C.A.; Damonte, E.B.; Rodriguez, J.B. Tetrahedron. 66(18):3332-3340
"Synthesis of PEGylated lactose analogs for inhibition studies on T.cruzi trans-sialidase" (2010) Giorgi, M.E.;Ratier, L.;Agusti, R. (...)De Lederkremer, R.M. Glycoconjugate Journal. 27(5):549-559
"Synthesis and GABAA receptor activity of A-homo analogues of neuroactive steroids" (2010) Dansey, M.V.;Di Chenna, P.H.;Veleiro, A.S. (...)Burton, G. European Journal of Medicinal Chemistry. 45(7):3063-3069
"2-C-Methyluridine modified hammerhead ribozyme against the estrogen receptor" (2010) Pontiggia, R.;Pontiggia, O.;Simian, M. (...)Iribarren, A.M. Bioorganic and Medicinal Chemistry Letters. 20(9):2806-2808
"10-23 DNAzyme modified with (2′R)- and (2′S)-2′-deoxy- 2′-C-methyluridine in the catalytic core" (2010) Robaldo, L.; Montserrat, J.M.; Iribarren, A.M. Bioorganic and Medicinal Chemistry Letters. 20(15):4367-4370
"Triterpenoids with acetylcholinesterase inhibition from chuquiraga erinacea D. Don. subsp. erinacea (Asteraceae)" (2010) Gurovic, M.S.V.;Castro, M.J.;Richmond, V. (...)Murray, A.P. Planta Medica. 76(6):607-610
"Enantiospecific synthesis of the sugar amino acid (2S,5S)-5-(aminomethyl)- tetrahydrofuran-2-carboxylic acid" (2010) Uhrig, M.L.; Simirgiotis, M.J.; Varela, O. Tetrahedron Asymmetry. 21(19):2435-2440
"Aeromonas hydrophila strains as biocatalysts for transglycosylation" (2010) Nbile, M.; Terreni, M.; Lewkowicz, E.; Iribarren, A.M. Biocatalysis and Biotransformation. 28(5-6):395-402
"Antiproliferative activity of synthetic naphthoquinones related to lapachol. First synthesis of 5-hydroxylapachol" (2010) Bonifazi, E.L.;Ríos-Luci, C.;León, L.G. (...)Misico, R.I. Bioorganic and Medicinal Chemistry. 18(7):2621-2630
"Allopregnanolone (3α-Hydroxy-5α-pregnan-20-one) derivatives with a polar chain in position 16α: Synthesis and activity" (2009) Slavíková, B.;Krištofíková, Z.;Chodounská, H. (...)Kasal, A. Journal of Medicinal Chemistry. 52(7):2119-2125
"Discovery of novel trichomonacidals using LDA-driven QSAR models and bond-based bilinear indices as molecular descriptors" (2009) Rivera-Barroto, O.M.;Marrero-Ponce, Y.;Meneses-Marcel, A. (...)Vogel, C. QSAR and Combinatorial Science. 28(1):9-26
"Structure-activity relationships of neuroactive steroids acting on the GABAA receptor" (2009) Veleiro, A.S.; Burton, G. Current Medicinal Chemistry. 16(4):455-472
"Highly stereoselective synthesis of steroidal 2,5-diketopiperazines based on isocyanide chemistry" (2009) Bruttomesso, A.C.; Eiras, J.; Ramírez, J.A.; Galagovsky, L.R. Tetrahedron Letters. 50(28):4022-4024
"Preparation and characterization of a novel starch-based interpolyelectrolyte complex as matrix for controlled drug release" (2009) Prado, H.J.; Matulewicz, M.C.; Bonelli, P.R.; Cukierman, A.L. Carbohydrate Research. 344(11):1325-1331
"Synthesis and evaluation of 1,1′-hydrocarbylenebis(indazol-3-ols) as potential antimalarial drugs" (2009) Alho, M.M.;García-Sánchez, R.N.;Nogal-Ruiz, J.J. (...)Arán, V.J. ChemMedChem. 4(1):78-87
"Synthesis of 9-β-d-arabinofuranosylguanine by combined use of two whole cell biocatalysts" (2009) Médici, R.; Iribarren, A.M.; Lewkowicz, E.S. Bioorganic and Medicinal Chemistry Letters. 19(15):4210-4212
"Synthesis and GABAA receptor activity of 2,19-sulfamoyl analogues of allopregnanolone" (2009) Durán, F.J.;Edelsztein, V.C.;Ghini, A.A. (...)Burton, G. Bioorganic and Medicinal Chemistry. 17(18):6526-6533
"Synthesis of pentopyranosyl-containing thiodisaccharides. Inhibitory activity against β-glycosidases" (2009) Cagnoni, A.J.; Uhrig, M.L.; Varela, O. Bioorganic and Medicinal Chemistry. 17(17):6203-6212
"Synthesis of 4-azasteroids by an intramolecular Ugi reaction" (2008) Alonso, F.; Acebedo, S.L.; Bruttomesso, A.C.; Ramírez, J.A. Steroids. 73(12):1270-1276
"Synthesis and evaluation of N-substituted acridones as antiviral agents against haemorrhagic fever viruses" (2008) Sepúlveda, C.S.;Fascio, M.L.;Mazzucco, M.B. (...)Damonte, E.B. Antiviral Chemistry and Chemotherapy. 19(1):41-47
"Synthesis and biological evaluation of 2-alkylaminoethyl-1,1-bisphosphonic acids against Trypanosoma cruzi and Toxoplasma gondii targeting farnesyl diphosphate synthase" (2008) Szajnman, S.H.;García Liñares, G.E.;Li, Z.-H. (...)Rodriguez, J.B. Bioorganic and Medicinal Chemistry. 16(6):3283-3290
"Anti-herpetic and anti-inflammatory activities of two new synthetic 22,23-dihydroxylated stigmastane derivatives" (2008) Michelini, F.M.;Ramírez, J.A.;Berra, A. (...)Alché, L.E. Journal of Steroid Biochemistry and Molecular Biology. 111(1-2):111-116
"New acridinone derivative with trypanocidal activity" (2008) Pardo Andreu, G.L.;Inada, N.M.;Pellón, R.F. (...)Vercesi, A.E. International Journal of Antimicrobial Agents. 31(5):502-504
"Nucleoside synthesis using a novel macroporous grafted polyethylene as biocatalyst support" (2008) Trelles, J.A.;Bentancor, L.;Grasselli, M. (...)Iribarren, A.M. Journal of Molecular Catalysis B: Enzymatic. 52-53(1-4):189-193
"Synthesis and antiviral activity of azoles obtained from carbohydrates" (2008) Barradas, J.S.;Errea, M.I.;D'Accorso, N.B. (...)Damonte, E.B. Carbohydrate Research. 343(14):2468-2474
"Synthesis of 1,3-oxazole and benzimidazole pendant groups from polyacrylonitrile hydrolysis products" (2008) Vega, I.N.; Sánchez, L.; D'Accorso, N. Journal of Heterocyclic Chemistry. 45(2):429-433
"Synthesis of novel carbohydrate acridinone derivatives with potential biological activities using 1,3-dipolar cycloaddition" (2007) Fascio, M.L.; D'Accorso, N.B.; Pellón, R.F.; Docampo, M.L. Synthetic Communications. 37(23):4209-4217
"An insight on targets and patented drugs for chemotherapy of chagas disease" (2007) Duschak, V.G.; Couto, A.S. Recent Patents on Anti-Infective Drug Discovery. 2(1):19-51
"Fluorine-containing aryloxyethyl thiocyanate derivatives are potent inhibitors of Trypanosoma cruzi and Toxoplasma gondii proliferation" (2007) Liñares, G.G.;Gismondi, S.;Codesido, N.O. (...)Rodriguez, J.B. Bioorganic and Medicinal Chemistry Letters. 17(18):5068-5071
"Preparation of potential 3-deazauridine and 6-azauridine prodrugs through an enzymatic alcoholysis" (2007) Zinni, M.A.; Iglesias, L.E.; Iribarren, A.M. Journal of Molecular Catalysis B: Enzymatic. 47(1-2):86-90
"Reduction of an amido zinc(II) phthalocyanine by diborane" (2006) Strassert, C.A.; Dicelio, L.E.; Awruch, J. Synthesis(5):799-802
"Antioxidant and antimicrobial activities of rosemary extracts linked to their polyphenol composition" (2006) Moreno, S.; Scheyer, T.; Romano, C.S.; Vojnov, A.A. Free Radical Research. 40(2):223-231
"Synthesis of 6-thia analogs of the natural neurosteroid allopregnanolone" (2006) Durán, F.J.; Ghini, A.A.; Coirini, H.; Burton, G. Tetrahedron. 62(20):4762-4768
"Nucleoside phosphorylases" (2006) Lewkowicz, E.S.; Iribarren, A.M. Current Organic Chemistry. 10(11):1197-1215
"Microbial synthesis of 2,6-diaminopurine nucleosides" (2006) Médici, R.; Lewkowicz, E.S.; Iribarren, A.M. Journal of Molecular Catalysis B: Enzymatic. 39(1-4):40-44
"Design, synthesis, and biological evaluation of phosphinopeptides against Trypanosoma cruzi targeting trypanothione biosynthesis" (2006) Ravaschino, E.L.; Docampo, R.; Rodriguez, J.B. Journal of Medicinal Chemistry. 49(1):426-435
"Synthesis of C(1)-C(11) oxygen-bridged pregnanes" (2005) Veleiro, A.S.;Taich, P.J.;Alvarez, L.D. (...)Burton, G. Tetrahedron Letters. 46(24):4235-4238
"Synthesis and biological evaluation of 1-amino-1,1-bisphosphonates derived from fatty acids against Trypanosoma cruzi targeting farnesyl pyrophosphate synthase" (2005) Szajnman, S.H.; Ravaschino, E.L.; Docampo, R.; Rodriguez, J.B. Bioorganic and Medicinal Chemistry Letters. 15(21):4685-4690
"Synthesis and antiviral evaluation of some carbonucleoside analogues" (2005) Martins Alho, M.A.;Errea, M.I.;Sguerra, V.L. (...)Damonte, E.B. Journal of Heterocyclic Chemistry. 42(5):979-983
"Antiviral mode of action of a synthetic brassinosteroid against Junin virus replication" (2005) Castilla, V.;Larzábal, M.;Sgalippa, N.A. (...)Coto, C.E. Antiviral Research. 68(2):88-95
"6,19-Sulfur-bridged progesterone analogues with antiimmunosuppressive activity" (2005) Veleiro, A.S.;Pecci, A.;Monteserín, M.C. (...)Burton, G. Journal of Medicinal Chemistry. 48(18):5675-5683
"Antiviral activity of natural and synthetic brassinosteroids" (2004) Wachsman, M.B.;Ramírez, J.A.;Talarico, L.B. (...)Coto, C.E. Current Medicinal Chemistry: Anti-Infective Agents. 3(2):163-179
"Benzimidazole as deazapurine analogue for microbial transglycosylation" (2004) Bentancor, L.;Trelles, J.A.;Nóbile, M. (...)Iribarren, A.M. Journal of Molecular Catalysis B: Enzymatic. 29(1-6):3-7
"Photochemistry of 2-acyloxycarbazoles. A potential tool in the synthesis of carbazole alkaloids" (2004) Bonesi, S.M.; Crevatín, L.K.; Erra-Balsells, R. Photochemical and Photobiological Sciences. 3(4):381-388
"Combination strategy using pure enzymes and whole cells as biocatalysts for the preparation of 2-hydroxyesters and lactones from 2-oxoglutaric acid" (2004) Rustoy, E.M.; Pereyra, E.N.; Moreno, S.; Baldessari, A. Tetrahedron Asymmetry. 15(23):3763-3768
"In vitro and in vivo antiherpetic activity of three new synthetic brassinosteroid analogues" (2004) Michelini, F.M.;Ramírez, J.A.;Berra, A. (...)Alché, L.E. Steroids. 69(11-12):713-720
"A solvent-free synthesis of coumarins using a Wells-Dawson heteropolyacid as catalyst" (2004) Romanelli, G.P.;Bennardi, D.;Ruiz, D.M. (...)Autino, J.C. Tetrahedron Letters. 45(48):8935-8939
"Lipase-catalyzed preparation of biologically active esters of dehydroepiandrosterone" (2004) Bruttomesso, A.C.; Tiscornia, A.; Baldessari, A. Biocatalysis and Biotransformation. 22(3):215-220
"Synthesis of 2-(pyrimidin-4-yl)indoles" (2003) Franco, L.H.; Palermo, J.A. Chemical and Pharmaceutical Bulletin. 51(8):975-977
"PhI=NSes mediated aziridination of 11-pregnane derivatives: Synthesis of an 11,12-aziridino analogue of neuroactive steroids" (2003) Di Chenna, P.H.;Dauban, P.;Ghini, A. (...)Dodd, R.H. Tetrahedron. 59(7):1009-1014
"Synthesis of anticonvulsant sulfamides. Theoretical study of the related mechanism" (2003) Gavernet, L.; Cisneros, H.S.; Bruno-Blanch, L.E.; Estiú, G.L. Theoretical Chemistry Accounts. 110(6):434-440
"Synthesis of conformationally locked carbocyclic nucleosides built on an oxabicyclo[3.1.0]hexane system" (2003) Comin, M.J.; Rodriguez, J.B.; Russ, P.; Marquez, V.E. Tetrahedron. 59(3):295-301
"Synthesis and GABAA receptor activity of a 6,19-oxido analogue of pregnanolone" (2003) Veleiro, A.S.;Rosenstein, R.E.;Jaliffa, C.O. (...)Burton, G. Bioorganic and Medicinal Chemistry Letters. 13(3):343-346
"Synthesis and isolation of chloro-β-carbolines obtained by chlorination of β-carboline alkaloids in solution and in solid state" (2003) Ponce, M.A.; Tarzi, O.I.; Erra-Balsells, R. Journal of Heterocyclic Chemistry. 40(3):419-426
"Synthesis and antiviral activity of sulfated and acetylated derivatives of 2β,3α-dihydroxy-5α-cholestane" (2003) Garrido Santos, G.A.;Murray, A.P.;Pujol, C.A. (...)Maier, M.S. Steroids. 68(2):125-132
"Oxido-bridged neurosteroid analogues. Synthesis of 2,19-oxido-allopregnanolone" (2003) Eduardo, S.L.; Ghini, A.A.; Burton, G. Arkivoc. 2003(10):468-476
"Pharmacophoric pattern of anti-epileptic sulfonamides and sulfamates. Theoretical study of the associated requirements" (2002) Barrios, I.A; Bruno-Blanch, L.E; Estiú, G.L Journal of Molecular Structure: THEOCHEM. 580(1-3):243-250
"Enantioselective synthesis of (+)-neplanocin F" (2002) Comin, M.J.; Leitofuter, J.; Rodríguez, J.B. Tetrahedron. 58(16):3129-3136
"Enzyme-catalyzed preparation of novel fatty acid derivatives of pyridoxine with surfactant activity" (2002) Baldessari, A.; Mangone, C.P. Biocatalysis and Biotransformation. 20(4):275-279
"Antiviral properties of natural and semi-synthetic compounds from Heliotropium filifolium resin " (2002) Torres, R.;Modak, B.;Urzúa, A. (...)Pujol, E.D.Y.C.A. Boletin de la Sociedad Chilena de Quimica. 47(3):259-263
"Synthesis, high-resolution NMR spectroscopic analysis, and single-crystal X-ray diffraction of isoxazoline tetracycles" (2002) Fascio, M.L.; Alvarez-Larena, A.; D'Accorso, N.B. Carbohydrate Research. 337(24):2419-2425
"An antiviral principle present in a purified fraction from Melia azedarach L. leaf aqueous extract restrains herpes simplex virus type 1 propagation" (2002) Alché, L.E.; Barquero, A.A.; Sanjuan, N.A.; Coto, C.E. Phytotherapy Research. 16(4):348-352
"Synthesis of (2′s)-2′-deoxy-2′-C-methylpurine nucleosides and their phosphoramidites" (2002) Caballero, G.; Gallo, M.; Montserrat, J.M.; Iribarren, A.M. Helvetica Chimica Acta. 85(5):1284-1294
"Design, synthesis, and biological evaluation of aryloxyethyl thiocyanate derivatives against Trypanosoma cruzi" (2002) Elhalem, E.;Bailey, B.N.;Docampo, R. (...)Rodriguez, J.B. Journal of Medicinal Chemistry. 45(18):3984-3999
"Synthesis of β-D-galactofuranosyl nucleoside analogues. A new type of β-D-galactofuranosidase inhibitor" (2001) Marino, C.; Herczegh, P.; De Lederkremer, R.M. Carbohydrate Research. 333(2):123-128
"One-pot biocatalyzed preparation of substituted amides as intermediates of pharmaceuticals" (2001) Baldessari, A.; Mangone, C.P. Journal of Molecular Catalysis - B Enzymatic. 11(4-6):335-341
"Preparation and cytotoxicity toward cancer cells of mono(arylimino) derivatives of β-lapachone" (2001) Di Chenna, P.H.;Benedetti-Doctorovich, V.;Baggio, R.F. (...)Burton, G. Journal of Medicinal Chemistry. 44(15):2486-2489
"Synthesis of novel alkylamino zinc(II) phthalocyanines" (2001) Rodríguez, M.E.; Strassert, C.A.; Awruch, J.; Dicelio, L.E. Journal of Heterocyclic Chemistry. 38(2):387-389
"Synthesis and properties of (2′S)- and (2′R)-2′-deoxy-2′-C-methyl oligonucleotides" (2001) Cicero, D.O.; Gallo, M.; Neuner, P.J.; Iribarren, A.M. Tetrahedron. 57(36):7613-7621
"Bisphosphonates derived from fatty acids are potent growth inhibitors of Trypanosoma cruzi" (2001) Szajnman, S.H.; Bailey, B.N.; Docampo, R.; Rodriguez, J.B. Bioorganic and Medicinal Chemistry Letters. 11(6):789-792
"A facile synthesis of 3-glycosyl-5-substituted-2-isoxazoles" (2001) Fascio, M.L.; D'Accorso, N.B. Synthetic Communications. 31(12):1913-1920
"Glycoinositolphospholipids, free and as anchors of proteins, in trypanosoma" (2001) de Lederkremer, R.M.; Bertello, L.E. Current Pharmaceutical Design. 7(12):1165-1179
"Synthesis and isolation of nitro-β-carbolines obtained by nitration of commercial β-carboline alkaloids" (2001) Ponce, M.A.; Erra-Balsells, R. Journal of Heterocyclic Chemistry. 38(5):1071-1082
"Acyclic analogues of deoxyadenosine 3',5'-bisphosphates as P2Y 1 receptor antagonists" (2000) Kim, Y.-C.;Gallo-Rodriguez, C.;Jang, S.-Y. (...)Jacobson, K.A. Journal of Medicinal Chemistry. 43(4):746-755
"Design and synthesis of aryloxyethyl thiocyanate derivatives as potent inhibitors of Trypanosoma cruzi proliferation" (2000) Szajnman, S.H.;Yan, W.;Bailey, B.N. (...)Rodriguez, J.B. Journal of Medicinal Chemistry. 43(9):1826-1840
"Enantiospecific synthesis of a glycoside of D-epi-purpurosamine" (2000) Iriarte Capaccio, C.A.; Varela, O. Tetrahedron Asymmetry. 11(24):4945-4954
"Synthesis and characterization of some N-heterocyclic carbohydrate derivatives" (2000) Alho, M.A.M.; D'Accorso, N.B. Molecules. 5(3):381-382
"Escherichia coli Bl21: A useful biocatalyst for the synthesis purine nucleosides" (2000) Rogert, M.C.;Martínez, N.;Porro, S. (...)Iribarren, A. Molecules. 5(3):535-536
"A simple enzymatic preparation of 2',3'-di-O-acetylnucleosides through a lipase catalyzed alcoholysis" (2000) Zinni, A.;Schmidt, A.;Gallo, M. (...)Iribarren, A. Molecules. 5(3):533-534
"Two approaches to the enantioselective synthesis of (4R)-(-)-4-hydroxymethyl-4-thiobutyro-1,4-lactone" (2000) Zunszain, P.A.; Varela, O. Tetrahedron Asymmetry. 11(3):765-771
"Synthesis of heterocylic compounds of biological interest from carbohydrate derivatives" (2000) Martinez Esperón, M.F.; Fascio, M.L.; D'Accorso, N.B. Molecules. 5(3):418-419
"Synthesis and characterization of 2,2-disubstituted thiadiazolines" (2000) Martins Alho, M.A.;Moglioni, A.G.;Brousse, B. (...)D'Accorso, N.B. Arkivoc. 2000(4 SPECISS):627-640
"Synthesis of aziridinosteroids" (2000) Di Chenna, P.;Dauban, P.;Ghini, A.A. (...)Dodd, R.H. Molecules. 5(3):443-444
"Synthesis of D-homo analogs of neurosteroids" (2000) Di Chenna, P.; Ghini, A.A.; Burton, G. Molecules. 5(3):447-448
"D-galactofuranosylphosphonates. First synthesis of UDP-C-D- galactofuranose" (1999) Kovensky, J.; McNeil, M.; Sinaÿ, P. Journal of Organic Chemistry. 64(17):6202-6205
"Synthesis of two isosteric phosphono analogues of D-galactofuranosyl phosphate" (1999) Kovensky, J.; Cirelli, A.F.; Sinay, P. Carbohydrate Letters. 3(4):271-276
"Synthesis of C-5'-nor-dideoxycarbanucleosides structurally related to neplanocin C" (1999) Comin, M.J.; Pujol, C.A.; Damonte, E.B.; Rodriguez, J.B. Nucleosides and Nucleotides. 18(10):2219-2231
"Synthesis and characterization of some nitrogen heterocycles from D- galactose derivatives" (1999) Faraco, A.A.G.;Prado, M.A.F.;D'Accorso, N.B. (...)Prado, R.F. Journal of Heterocyclic Chemistry. 36(5):1129-1133
"Enantioselective synthesis of (2R,4S)- and (2S,4R)-4-hydroxypipecolic acid from D-glucoheptono-1,4-lactone" (1999) Di Nardo, C.; Varela, O. Journal of Organic Chemistry. 64(17):6119-6125
"1-Thio-β-D-galactofuranosides: Synthesis and evaluation as β-D-galactofuranosidase inhibitors" (1998) Marino, C.;Mariño, K.;Miletti, L. (...)De Lederkremer, R.M. Glycobiology. 8(9):901-904
"Straightforward synthesis of a derivative of purpurosamine C from D- galactose" (1998) Zunszain, P.A.; Varela, O. Tetrahedron Asymmetry. 9(7):1269-1276
"Stereospecific synthesis of steroidal 20,16-γ-carbolactones" (1998) Bruttomesso, A.C.; Doller, D.; Gros, E.G. Synthetic Communications. 28(21):4043-4057
"Structure-activity relationship of new growth inhibitors of Trypanosoma cruzi" (1998) Cinque, G.M.;Szajnman, S.H.;Zhong, L. (...)Gros, E.G. Journal of Medicinal Chemistry. 41(9):1540-1554
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"Synthesis of [131-I]-iodinated quercetin" (1997) Barolli, M.G.; Pomilio, A.B. Journal of Labelled Compounds and Radiopharmaceuticals. 39(11):927-933
"Synthesis of 131I derivatives of indolealkylamines for brain mapping" (1997) Sintas, J.A.; Vitale, A.A. Journal of Labelled Compounds and Radiopharmaceuticals. 39(8):677-684
"Anomalous Horner-Wadsworth-Emmons reactions on 3,4-enuloses" (1997) Moradei, O.M.; Du Mortier, C.M.; Cirelli, A.F. Tetrahedron. 53(22):7397-7402
"Synthesis and photophysical properties of a new cationic water-soluble Zn phthalocyanine" (1997) Fernández, D.A.; Awruch, J.; Dicelio, L.E. Journal of Photochemistry and Photobiology B: Biology. 41(3):227-232
"Facile synthesis of glycofuranosyl isothiocyanates" (1997) Marino, C.; Varela, O.; De Lederkremer, R.M. Carbohydrate Research. 304(3-4):257-260
"Conversion of benzaldehyde into benzyl benzoate from the reaction with lithium metal in hexane" (1997) Nudelman, N.S.; Mendiara, S. Tetrahedron Letters. 38(13):2245-2248
"Stereocontrolled synthesis of stereoregular, chiral analogs of nylon 5,5 and nylon 5,6" (1997) Orgueira, H.A.; Varela, O. Tetrahedron Asymmetry. 8(9):1383-1389
"Gemini surfactants from alkyl glucosides" (1997) Castro, M.J.L.; Kovensky, J.; Fernández Cirelli, A. Tetrahedron Letters. 38(23):3995-3998
"Synthesis of oxido-bridged analogs of 18-hydroxyprogesterone" (1996) Benedetti Doctorovich, M.O.V.; Ghini, A.A.; Burton, G. Steroids. 61(6):345-348
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"Kinetics and mechanism of the heterogeneous oxidation of ethane and ethylene on samarium(III) oxide" (1996) Amorebieta, V.T.; Colussi, A.J. Journal of the American Chemical Society. 118(42):10236-10241
"86. Lipase-catalysed regioselective deacetylation of androstane derivatives" (1996) Baldessari, A.; Bruttomesso, A.C.; Gros, E.G. Helvetica Chimica Acta. 79(4):999-1004
"Ring expansion of fused cyclopropylketones. Synthesis of a 12(13→18)-abeo-pregnane" (1996) Ferrara, A.; Burton, G. Tetrahedron Letters. 37(7):929-932
"Ritter reaction on terpenoids. IV. Remarkable tendency to produce 3-aza-bicyclo[3.3.1]non-2-ene systems from mono and sesquiterpenes" (1995) Rodriguez, J.B.; Gros, E.G.; Caram, J.A.; Marschoff, C.M. Tetrahedron Letters. 36(43):7825-7828
"Reduction of a Δ4-Steroid with Diborane" (1995) D'Alessandro, C.; Giacopello, S.; Seldes, A.M.; Deluca, M.E. Synthetic Communications. 25(18):2703-2708
"Preparation and biological evaluation of technetium‐99m‐phenylethylamine complexes" (1995) Vitale, A.A.;Calvino, M.A.;Ferrari, C.C. (...)Pomilio, A.B. Journal of Labelled Compounds and Radiopharmaceuticals. 36(6):509-519
"Syntheses of 21-hydroxy-11,19-oxidopregn-4-ene-3,20-dione and 21-hydroxy-6,19-oxidopregn-4-ene-3,20-dione" (1995) Veleiro, A.S.; Nevado, M.V.; Monteserín, M.C.; Burton, G. Steroids. 60(3):268-271
"Synthesis of some oxadiazole derivatives of d‐mannose" (1995) Fascio, M.L.; D'Accorso, N.B. Journal of Heterocyclic Chemistry. 32(3):815-818
"Cleavage of acetals promoted by copper (II) sulphate adsorbed on silica gel" (1995) Caballero, G.M.; Gros, E.G. Synthetic Communications. 25(3):395-404
"Synthesis of 4-methylcoumarin-7-yl β-d-galactofuranoside, a fluorogenic substrate for galactofuranosidase" (1995) Marino, C.; Cancio, M.J.; Varela, O.; de Lederkremer, R.M. Carbohydrate Research. 276(1):209-213
"Design, synthesis, and anti‐ Trypanosoma cruzi evaluation of a new class of cell‐growth inhibitors structurally related to Fenoxycarb" (1995) Schvartzapel, A.J.;Fichera, L.;Esteva, M. (...)Gros, E.G. Helvetica Chimica Acta. 78(5):1207-1214
"Synthetic reactions of aldonolactones" (1994) De Lederkremer, R.M.; Varela, O. Advances in Carbohydrate Chemistry and Biochemistry. 50(C):125-209
"The first synthesis of an A-ring fused steroidal isothiazole" (1994) Giacopello, S.; Deluca, M.E.; Seldes, A.M. Tetrahedron Letters. 35(36):6643-6646
"A short synthesis of (2S,4S,5R)-4,5,6-trihydroxynorleucine" (1994) Varela, O.; Nin, A.P.; De Lederkremer, R.M. Tetrahedron Letters. 35(50):9359-9362
"Starfish saponins, Part 2. Steroidal oligoglycosides from the starfish cosmasterias lurida" (1994) Roccatagliata, A.J.;Maier, M.S.;Seldes, A.M. (...)Minale, L. Journal of Natural Products. 57(6):747-754
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"Synthesis of [20,21‐13C2]‐pregnenolone" (1993) Caballero, G.M.; Gros, E.G. Journal of Labelled Compounds and Radiopharmaceuticals. 33(10):907-911
"Synthesis and antitumor activity of anthracycline disaccharide glycosides containing daunosamine" (1993) Horton, D.; Priebe1, W.; Sznaidmanc, M.L.; Varela, O. Journal of Antibiotics. 46(11):1720-1730
"Synthesis of 14C‐(carbonyl)‐N‐(4‐iodo‐2,6‐diethylphenylcarbamoylmethyl)‐iminodiacetic acid" (1993) Pozzi, O.R.; Arciprete, C.P.; Gros, E.G.; Mitta, A.E.A. Journal of Labelled Compounds and Radiopharmaceuticals. 33(4):259-262
"Diastereoselective synthesis of cis-4-hydroxypipecolic acid from D-glucosamine." (1993) Nin, A.P.; Varela, O.; de Lederkremer, R.M. Tetrahedron. 49(42):9459-9464
"Preparation and Biological Activities of Sulfated Derivatives of (1→3)-β-D-Glucans" (1991) Suzuki, T.;Ohno, N.;Adachi, Y. (...)Yadomae, T. Journal of Pharmacobio-Dynamics. 14(5):256-266
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"Synthesis of |21‐14C|‐3β‐hydroxy‐5β‐pregnan‐20‐one and |21‐14C|‐5β‐cholestan‐3β‐ol" (1985) Garraffo, H.M.; Deluca, M.E.; Seldes, A.M.; Gross, E.G. Journal of Labelled Compounds and Radiopharmaceuticals. 22(7):673-676
"Preparation of 3β -Acetoxy-5β-pregnan-20-one from 3 a- Acetoxy-5β-cholan-24-oic Acid Aimed at the Isotopic Labelling of the Pregnane Side Chain" (1984) Deluca, M.E.; Seldes, A.M.; Garraffo, H.M.; Gros, E.G. Zeitschrift fur Naturforschung - Section B Journal of Chemical Sciences. 39(11):1617-1621
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"A new approach to the synthesis of 3β,23-diacetoxy-24-nor-5-cholene from 3β,21-diacetoxy-5-pregnen-20-one" (1980) Seldes, A.M.; Anding, C.R.; Gros, E.G. Topics in Catalysis. 36(5):575-580
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